Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking

Authors: Xiaobo Wan, Tangpo Yang, Adolfo Cuesta, Xiaming Pang, Trent E. Balius, John J. Irwin, Brian K. Shoichet, Jack Taunton

Published: 2020-02-27

DOI: 10.1021/jacs.9b10377

Source: Full article


Abstract

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