Abstract 1657: Discovery of a first-in-class multifunctional TYMS non-classical antifolate inhibitors with potent <i>in vivo</i> activity that prolongs survival

Authors: Peter Elias Dib, Maria Guijarro, Patrick Kellish, Nick Paciaroni, Akbar Nawab, Jacob Andring, Lidia Kulemina, Derek Leas, Nick Borrero, Carlos Modenutti, Richard Bennett, Jonathan Licht, Robert McKenna, Adrian Roitberg, Frederic Kaye, Maria Zajac-Kaye

Published: 2023-04-04

DOI: 10.1158/1538-7445.am2023-1657

Source: Full article


Abstract

Abstract