Abstract 3428: Discovery of a highly potent and selective dual PROTAC degrader of CDK12 and CDK13

Authors: Yu Chang, Jianzhang Yang, Jean Ching-Yi Tien, Zhen Wang, Yang Zhou, Pujuan Zhang, Weixue Huang, Josh Vo, Ingrid J. Apel, Cynthia Wang, Victoria Zhixuan Zeng, Yunhui Cheng, Shuqin Li, George Xiaoju Wang, Ke Ding, Arul M. Chinnaiyan

Published: 2023-04-04

DOI: 10.1158/1538-7445.am2023-3428

Source: Full article


Abstract

Abstract