Authors: Wai Cheung Chan, Shabnam Sharifzadeh, Sara J. Buhrlage, Jarrod A. Marto
Published: 2021-06-18
DOI: 10.1039/d1cs00231g
Source: Full article
The past decade has witnessed growing enthusiasm for covalent drug discovery. We review foundational and cutting-edge mass spectrometry chemoproteomic methods for covalent drug discovery: target ID, hit discovery, and lead characterization.