What a difference a methylene makes: replacing Glu with Asp or Aad in the Lys-urea-Glu pharmacophore of PSMA-targeting radioligands to reduce kidney and salivary gland uptake
Authors: Hsiou-Ting Kuo, Kuo-Shyan Lin, Zhengxing Zhang, Chengcheng Zhang, Helen Merkens, Ruiyan Tan, Aron Roxin, Carlos F. Uribe, François Bénard